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Kristoffer Sahlholm
Kontakt
E-post
kristoffer.sahlholm@umu.se
Telefon
090-786 67 77
Verksam vid
Anknytning
Universitetslektor vid
Institutionen för medicinsk och translationell biologi
Enhet: Grupp Kristoffer Sahlholm, Lärare D1-flygeln
Plats
hus H, Johan Bures väg 12, Biologihuset
Umeå universitet, 901 87 Umeå
Anknytning
Anknuten som övrig/annan befattning till
Wallenberg centrum för molekylär medicin vid Umeå universitet (WCMM)
Plats
Umeå universitet, 901 87 Umeå
Publikationer
Publikationer
Forskning
Forskning
2024
Neurophysiological treatment effects of mesdopetam, pimavanserin and clozapine in a rodent model of Parkinson's disease psychosis
Neurotherapeutics
, Elsevier 2024, Vol. 21, (2)
Stan, Tiberiu Loredan; Ronaghi, Abdolaziz; Barrientos, Sebastian A.; et al.
2023
Dopamine-induced arrestin recruitment and desensitization of the dopamine D4 receptor is regulated by G protein-coupled receptor kinase-2
Frontiers in Pharmacology
, Frontiers Media S.A. 2023, Vol. 14
Burström, Viktor; Ågren, Richard; Betari, Nibal; et al.
2023
Remote local photoactivation of morphine produces analgesia without opioid-related adverse effects
British Journal of Pharmacology
, John Wiley & Sons 2023, Vol. 180, (7) : 958-974
López-Cano, Marc; Font, Joan; Aso, Ester; et al.
2023
Unique effect of clozapine on adenosine A
2A
-dopamine D
2
receptor heteromerization
Biomedicine and Pharmacotherapy
, Elsevier 2023, Vol. 160
Valle-León, Marta; Casajuana-Martin, Nil; del Torrent, Claudia Llinas; et al.
2023
In vitro comparison of ulotaront (SEP-363856) and ralmitaront (RO6889450): two TAAR1 agonist candidate antipsychotics
International Journal of Neuropsychopharmacology
, Oxford University Press 2023, Vol. 26, (9) : 599-606
Ågren, Richard; Betari, Nibal; Saarinen, Marcus; et al.
2023
An E280K Missense Variant in KCND3/Kv4.3—Case Report and Functional Characterization
International Journal of Molecular Sciences
, MDPI 2023, Vol. 24, (13)
Ågren, Richard; Geerdink, Niels; Brunner, Han G.; et al.
2023
Major genetic risk factors for Dupuytren's disease are inherited from neandertals
Molecular biology and evolution
, Oxford University Press 2023, Vol. 40, (6)
Ågren, Richard; Patil, Snehal; Zhou, Xiang; et al.
2022
TAAR1 dependent and independent actions of the potential antipsychotic and dual TAAR1/5-HT1A receptor agonist SEP-383856
Neuropsychopharmacology
, Springer Nature 2022, Vol. 47 : 2319-2329
Saarinen, Marcus; Mantas, Ioannis; Flais, Ivana; et al.
2022
Evidence for two modes of binding of the negative allosteric modulator SB269,652 to the dopamine D2 receptor
Biomedicines
, MDPI 2022, Vol. 10, (1)
Ågren, Richard; Sahlholm, Kristoffer
2021
Synthetic corticosteroids as tryptophan hydroxylase stabilizers
Future Medicinal Chemistry
, Future Science Ltd. 2021, Vol. 13, (17) : 1465-1474
Betari, Nibal; Teigen, Knut; Sahlholm, Kristoffer; et al.
2021
Interaction of ligands for pet with the dopamine d3 receptor: in silico and in vitro methods
Biomolecules
, MDPI 2021, Vol. 11, (4)
Hsieh, Chia-Ju; Riad, Aladdin; Lee, Ji Youn; et al.
2021
V374A KCND3 Pathogenic Variant Associated With Paroxysmal Ataxia Exacerbations
Neurology Genetics
, American Academy of Neurology 2021, Vol. 7, (1)
Paucar, Martin; Ågren, Richard; Li, Tianyi; et al.
2021
Mechanistic insights into dopaminergic and serotonergic neurotransmission: concerted interactions with helices 5 and 6 drive the functional outcome
Chemical Science
, Royal Society of Chemistry 2021, Vol. 12, (33) : 10990-11003
Stepniewski, Tomasz Maciej; Mancini, Arturo; Ågren, Richard; et al.
2021
Decreased striatal adenosine A
2A
-dopamine D
2
receptor heteromerization in schizophrenia
Neuropsychopharmacology
, Springer Nature 2021, Vol. 46 : 665-672
Valle-Leon, Marta; Callado, Luis F.; Aso, Ester; et al.
2021
G protein-coupled receptor kinase-2 confers isoform-specific calcium sensitivity to dopamine D
2
receptor desensitization
The FASEB Journal
, John Wiley & Sons 2021, Vol. 35, (11)
Ågren, Richard; Sahlholm, Kristoffer
2021
Dopamine d
2
receptor agonist binding kinetics: role of a conserved serine residue
International Journal of Molecular Sciences
, MDPI 2021, Vol. 22, (8)
Ågren, Richard; Stepniewski, Tomasz Maciej; Zeberg, Hugo; et al.
2020
Discovery and biological characterization of a novel scaffold for potent inhibitors of peripheral serotonin synthesis
Future Medicinal Chemistry
, Future Science 2020, Vol. 12, (16) : 1461-1474
Betari, Nibal; Sahlholm, Kristoffer; Ishizuka, Yuta; et al.
2020
Inhibition of Tryptophan Hydroxylases and Monoamine Oxidase-A by the Proton Pump Inhibitor, Omeprazole-In Vitro and In Vivo Investigations
Frontiers in Pharmacology
, Frontiers Media S.A. 2020, Vol. 11
Betari, Nibal; Sahlholm, Kristoffer; Morato, Xavier; et al.
2020
A Neanderthal Sodium Channel Increases Pain Sensitivity in Present-Day Humans
Current Biology
, Elsevier 2020, Vol. 30, (17) : 3465-3469
Zeberg, Hugo; Dannemann, Michael; Sahlholm, Kristoffer; et al.
2020
Voltage-Dependent Dopamine Potency at D-1-Like Dopamine Receptors
Frontiers in Pharmacology
, Frontiers Media S.A. 2020, Vol. 11
Ågren, Richard; Sahlholm, Kristoffer
2020
Ligand with Two Modes of Interaction with the Dopamine D-2 Receptor-An Induced-Fit Mechanism of Insurmountable Antagonism
ACS Chemical Neuroscience
, American Chemical Society (ACS) 2020, Vol. 11, (19) : 3130-3143
Ågren, Richard; Zeberg, Hugo; Stępniewski, Tomasz Maciej; et al.
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